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Cardiac Treatment What are 3 treatments for heart disease? Treatment Cholesterol drugs. Medications can help lower bad cholesterol and reduce plaque buildup in the arteries. ... Aspirin. ... Beta blockers. ... Calcium channel blockers. ... Angiotensin-converting enzyme (ACE) inhibitors and angiotensin II receptor blockers (ARBs). ... Nitroglycerin. ... Ranolazine.